Basic Peptide Information

DICL ID
DICL_Pep_03854
Ion Channel
Neuronal acetylcholine receptor subunit alpha-4/beta-2
Peptide Function
Inhibitor
Gene Name
CHRNA4/CHRNB2

Activity Data (nM)

IC50
152 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
IRDγCCSNPACRVNNOHVC
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
GID
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
pH 7.1 to 7.5
Holding Potential (mV)
−70 mV
Temperature
Not mention
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available